New polymer teknolojia inoita kuti pave nechepamusoro peganda rakanaka
Zvose zvitsva zvinogadzirwa kana kuti kubudirira mune imwe nzira zvinokonzera mavambo acho kune basa revamwe. Mishonga mitsva uye mishonga miviri yemishonga haisi yakasiyana. Kana iwe uchikwanisa kuvandudza pane zvakagadzirwa neumwe musayendisiti, uye kufambira mberi kwako kwakanyatsobudirira, zviri nyore uye zvakachengeteka, iwe unenge uri pane chimwe chinhu.
Munguva ichangopfuura, dzakawanda zvehupomberi dzakapoteredza nhau dzeimwe itsva ibuprofen ganda rakagadzirwa nevanotsvakurudza paYunivhesiti yeWarwick pamwe nekambani yavo inobatsira Medherant.
Sezviri pachena, iyi patch delivery system inonyanya kukosha, isingasviki uye inopa mishonga yakawanda zvakanyanya kupfuura chero chinhu chatinenge tisina kumira pamitumbi yedu.
Ibuprofen Chii?
Ibuprofen (funga Advil kana Motrin) inonzi NSAID (nonsteroidal anti-inflammatory drug) iyo inobvumira inhibits cyclooxygenase-1 (COX-1) uye cyclooxygenase-2 (COX-2) enzyme saka inopesana neprogaglandin yekugadzirwa. Nokupindira ne prostaglandin synthesis, ibuprofen inobatsira kuderedza marwadzo, kupisa uye fivha. Zvinyorwa, dzimwe NSAID dzinosanganisira aspirin uye naproxen.
Nyanzvi dzinofungidzira kuti kunze kwekuvhiringidza prostaglandin yekugadzira, ibuprofen inogonawo kurwisa kuvhiringidza kuburikidza neropa mukati mune dzimwe nzira, kusanganisira kuchinjwa kwemuitiro we lymphocyte, kuvharwa kwekemotaxis, kuvhara kwe-neutrophil aggregation kana kushandiswa, uye kuderera kwezvinoshandiswa neproinflammatory cytokine levels.
Chii Ibuprofen Inoshandiswa?
Ibuprofen inoshandiswa kuderedza fivhiri pamwe nekubata zvirwere zvakasiyana-siyana uye marwadzo, zvakadai seaya anokonzerwa nemusoro wepamusoro, kudzoka shure, arthritis, manyowa uye nguva yekuenda kumwedzi.
Zvinofadza kuti NSAIDs seybuprofen zvakanyatsonaka pakurapa marwadzo eminyo. Uyezve, ibuprofen inogona kusanganiswa neopioid (yakadai sehydrocodone) kuti iite marwadzo akawanda.
Ibuprofen Inotungamirirwa Sei?
Nzira dzakasiyana-siyana dzehutongi dziripo kune ibuprofen, kusanganisira mapiritsi, injection, uye gels.
Kutungamirirwa kweIbuprofen kuburikidza nechigamba chinhu chitsva uye zviri nani pane zvinyorwa zvekushandisa shandisa gel. Ibuprofen gels zvinosvibisa uye haasi kuzorapa mishonga nguva dzose.
Heano mamwe mazano anofungidzirwa eIbuprofen patch uye yakanyanyisa po polymer teknolojia:
- Inyanzvi itsva inobvumira kuti chikwata chiremerwe nemaminitsi mashanu kana gumi mamwe mishonga. Mune mamwe mazwi, 30 muzana yehutachiwana hwechikwata chiri chaiyo mishonga.
- Kusunungurwa kwemishonga mumuviri kunowedzera kushanda uye kunogona kushanda kusvika maawa gumi nemaviri. Pari zvino, vanhu vane madhoji makuru eIbuprofen vangada kuedza mapiritsi maawa mana.
- Iyo chikwata chinonyanya kuomesa, kushanduka, kusununguka uye kutonhora kupfuura mamwe mavara. Uyezve, chigamba chinosiya zvishoma uye zvakasara uye zvakajeka.
Ibuprofen patch yakagadzirwa kushandiswa kwema polymer teknolojia yakagadzirirwa nekambani inonzi Bostik uye ine mvumo yekushandiswa kwemutambo neMedherant.
Zvimwe Zvichida Applications zvePatch Patsva Zvingave Zvine Mhepo-Kuchinja
Maererano neMedherant, dzakawanda dzemarwadzo-matanho ekuzorora ayo aripo panguva ino haaine peinkiller mishonga uye pane kusunungura kupisa (kufunga menthol). Nokudaro, izvi zvipfeko zvekare zvakaderera mukushandiswa kwavo. Nhamba itsva yeMedherant ibuprofen patch inogadzirwa nenzira dzakasiyana-siyana.
Chokutanga nokuti chikwata chacho hachizivikanwi, kwenguva yakareba-kuita uye nyore nyore kushandisa, inogona kunyatsobatsira kune vamwe varwere vanoita sevatambi uye vanhu vanorwara nemishonga yekuteerera . Semuenzaniso, mutambi angashandisa chigamba kune imwe nzvimbo yekushungurudzika kana kushandiswa kwemaawa, kana munhu ari kuverenga mishonga yakawanda anogona kunge asina mapiritsi maduku kuti azvidye pamusoro.
Chechipiri, kuburikidza nekupedza mudumbu uye kusunungura mishonga zvakananga kuburikidza neganda, ibuprofen patch inogona kuita kuti musikana usagumburwa, zvinowanzova nengozi kune avo vane mahombekiti akawandisa emakondomu eNSAID.
Chechitatu, teknolojia inoshandiswa kukudziridza chigamba ichi inogona kusarudzwa kuunza mamwe mishonga yemishonga-mishonga, iyo yakafanana neIbuprofen, yakanga isina kumbogadziriswa kuisa purogiramu. Nezvimwewo, zvinorwadza zvinorwadza zvinoshandiswawo patch form sezvakaitwa fentanyl (anpipiid) uye lidocaine (antichetic anesthetic), uye zvingava zvinonakidza kuona kana chigadzirwa ichi chitsva chinogona kuvandudza kutungamirirwa kwemishonga iyi, zvakare.
Ibuprofen Inobatsira Zvikuru Here?
Ibuprofen inotengeswa pamusoro pekambani uye njodzi yemigumisiro yakaipa yakaderera. Kusuruvara kwepamuviri ndiko kunonyanya kukanganiswa kweASAID seybuprofen. Imwe mimwe migumisiro yakaipa yeIbuprofen inosanganisira kubuda ropa (kufanana neuropi inopa ropa kana kuti kurohwa) uye kushungurudzwa kwesonda.
Tarisa nyaya ino pamusoro pekuti NSAIDs dzinobatanidzwa sei kune ma testes asina kufanira mucheche.
Sezvambotaurwa, vaiti vehutsva ibuprofen patch vanoti nechikafu chavo, hapana ngozi yekurwadziwa kwepamuviri nokuti mishonga inobatwa neganda kwete nehutachiona.
Zvisinei, pane zvisingawanzoitiki, ibuprofen inogona kukonzera kusvibiswa kwakashata, mikoko uye mamwe maitiro eganda. Vanhu vane nhoroondo yeatopy , kana avo vane "hyperallergic" uye vanotambura kubva kune eczema, hay fever uye inokonzerwa nechirwere chemafi, inowanzove yeropaji kune ibuprofen. Kunyange zvakadaro, vanhu vasina nharaunda vakagadzirisa zvirwere zvese kuIbuprofen.
Ibuprofen patch iri kure kure nekurova pamusika uye haichiri kuva FDA inogamuchirwa. Kusvika ikozvino, pane zvishoma zvitsvakurudzo zvakabudiswa pachikwata-zvizhinji zvatinoziva zvinouya kubva kumashizha ekubudisa, kubvunzurudzwa uye mharidzo dzevhidhiyo-uye isu tichada kuona zvimwe zvakadzama data tisati tanyatsonzwisisa uku kuumbwa patsva. Semuenzaniso, izvo zvisinganzwisisiki kana kuwedzera kwemazi uye zvakasimudzirwa kwemashoko ekubudirira kweibuprofen patch zvingangoita kuti kuwedzera kweganda kuve kune avo vanokonzerwa neNSAIDs.
Kutarisa mberi, Medherant, muiti we ibuprofen patch, anotarisira kuti ino rivhi-drug-delivery system iyo inoshandiswa kugadzirisa mamwe mishonga uye pamusoro-the-counter painkillers dzakawanda dzakanga dzisati dzawanikwa musina chigamba. Somuenzaniso, Medherant iri kuedza nemethyl salicylate patch. (Methly salicylate ndiyo inonyanya kushandiswa muBENGAY.)
Sources
Chinyorwa chinonzi "Delayed-type hypersensitivity rash kubva kuIbuprofen" neE Nettis uye vanyori vanyori vakaparidzirwa muAirergy muna 2003.
Muchikamu chinonzi "Ibuprofen" kubva kuDrug Monographs chikamu che Access Access.